Soo saaraha budada Amino Tadalafil Lambarka CAS: 385769-84-6 98% daahirnimo ugu yaraan maaddooyinka dheeraadka ah
Fiidiyowga Badeecada
Cabbiraadaha Badeecada
| Magaca alaabta | Amino Tadalafil |
| Magac kale | (6R,12aR)-2-Amino-6-(1,3-benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4-dione;AminoTadalafil(6R,12Ar)-2-Amino-6-(1,3-Benzodioxol-5-Yl)-2,3,6,7,12,12A-Hexahydropyrazino[1',2':1,6]Pyrido[3,4-B]Indole-1,4-Dion e;(6R,12aR)-2-Amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,6,7,12,12a-hexahydropyrazino[1',2':1,6]pyrido[3,4-b]indol-1,4-dione;(6R,12aR)-2-amino-6-(benzo[d][1,3]dioxol-5-yl)-2,3,12,12a-tetrahydropyrazino[1',2':1,6]pyrido[3,4-b]indole-1,4(6H,7H)-dione |
| Lambarka CAS. | 385769-84-6 |
| Qaacidada moolikaalka | C21H18N4O4 |
| Miisaanka molecular-ka | 390.39 |
| Daahirnimo | 98.0% |
| Muuqaalka | Budada cad ilaa budo cad |
| Codsiga | Qalabka Cuntada ee Cayriin ah |
Soo bandhigida badeecada
Amino Tadalafil waa iskudhis cusub, oo ka soo jeeda tadalafil, kaas oo si isa soo taraysa caan uga noqonaya goobta cillad kacsiga (ED). Waxay isku daraysaa amino acid-ka iyo tadalafil, oo ah daawo ka hortagta PDE5 oo ay FDA ansixisay oo inta badan loo isticmaalo daawaynta ED. Waxay ka shaqaysaa kordhinta socodka dhiigga ee guska, taasoo u oggolaanaysa ragga inay gaaraan oo ay ilaaliyaan kacsiga. Dhanka kale, amino acids-ku waxay door muhiim ah ka ciyaaraan hawlaha kala duwan ee jirka, oo ay ku jiraan soo saarista borotiinnada, kuwaas oo ah qaybaha dhismaha unugyada iyo xubnaha. Isku-darka labadan maaddooyin waxaa loogu talagalay in lagu xoojiyo waxtarka Tadalafil ee daaweynta ED. Amino Tadalafil waa nooc la hagaajiyay oo leh awood aan caadi ahayn, taasoo kor u qaadaysa waxqabadka iyo kala-duwanaanta kii ka horreeyay. Qaab-dhismeedkeeda kiimikada ayaa weli la mid ah Tadalafil, laakiin iyada oo loo marayo soo bandhigidda kooxaha amino, waxay heshaa tayooyin gaar ah oo ka dhigaya inay ka soo muuqato adduunka dawooyinka. Sida tadalafil, Amino Tadalafil waxay ka shaqeysaa joojinta phosphodiesterase 5 (PDE5), enzyme-ka mas'uulka ka ah jebinta guanosine monophosphate (cGMP) ee jirka. cGMP waa isku-dhis dabiici ah oo kor u qaada nasashada xididdada dhiigga, taasoo kordhisa socodka dhiigga. Iyada oo la joojinayo PDE5, amino Tadalafil waxay hubisaa ururinta cGMP, taasoo kor u qaadaysa vasodilation-ka iyo hagaajinta wareegga dhiigga. Intaa waxaa dheer, cilmi-baarayaashu waxay sahamiyeen awooddeeda ay ku caawin karto daaweynta benign prostatic hyperplasia (BPH) iyadoo kor u qaadaysa socodka dhiigga ee qanjirka 'prostate'.
Muuqaalka
(1) Nadiifnimo sare: Amino Tadalafil waxay heli kartaa badeecooyin saafi ah iyada oo loo marayo hababka wax soo saarka ee sifeynta. Nadiifnimo sare waxay ka dhigan tahay helitaan wanaagsan oo noolaha ah iyo falcelin xun oo yar.
(2) Badbaadada: Badbaado sare, falcelin xun oo yar.
(3) Xasillooni: Amino Tadalafil waxay leedahay xasillooni wanaagsan waxayna ilaalin kartaa firfircoonideeda iyo saameynteeda iyadoo la raacayo jawiyo iyo xaalado kaydin oo kala duwan.
Codsiyada
Amino Tadalafil waa daawo ka hortagta PDE5 oo leh saameyn daawo oo la mid ah tadalafil. Iyadoo la isku darayo amino acids iyo tadalafil, amino Tadalafil waxaa loo maleynayaa inuu ka waxtar badan yahay daaweynta cillad kacsiga marka loo eego tadalafil oo keliya. Amino acid waxay gacan ka geysan kartaa kor u qaadista wareegga dhiigga waxayna taageeri kartaa waxtarka guud ee daawooyinka. Intaa waxaa dheer, waxay hagaajin kartaa calaamadaha cillad kacsiga (ED) iyadoo xannibaysa dhaqdhaqaaqa enzyme-ka PDE5 si kor loogu qaado socodka dhiigga ee xubnaha taranka ragga. Marka la barbardhigo tadalafil, amino Tadalafil si tartiib tartiib ah ayaa loogu dheefshiidaa jirka waxayna soo saari kartaa saameyn waarta. Tani waxay siineysaa amino Tadalafil awood weyn oo lagu daaweynayo ED.












