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Soo saaraha budada Nefiracetam CAS No.: 77191-36-7 99% nadiifinta min.maaddooyinka dheeriga ah

Sharaxaad Gaaban:

Nefiracetam waxay ka tirsan tahay fasalka kobcinta sirdoonka aan xuduudka lahayn ee daroogada, kuwaas oo leh qaabab kiimiko oo kala duwan oo kor u qaadaya awoodda garashada iyo ka hortagga dhaawaca barashada iyo xusuusta iyada oo loo marayo saamaynta ay ku leeyihiin kiliyaha maskaxda.


Faahfaahinta Alaabta

Tags Product

Qiyaasta Alaabta

Magaca alaabta

Nefiracetam

Magac kale

n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamide; NEFIRACETAM;

2-oxo-1-pyrrolidinylaceticacid,2,6-dimethylanilide;

dm9384;

n- (2,6-dimethylphenyl) -2-oxo-1-pyrrolidineacetamid; DM-9384, (2- (2-Oxopyrrolidin-1-yl) -N- (2,6-dimethylphenyl) -acetamide;

DMPA

CAS Maya.

77191-36-7

qaacidada molecular

C14H18N2O2

Miisaanka molecular

246.3

daahirnimo

99.0%

Muuqashada

budo cad

Baakad

25 kg / foosto

Codsiga

nootropic

hordhaca alaabta

Nefiracetam waxay ka tirsan tahay fasalka kobcinta sirdoonka aan xuduudka lahayn ee daroogada, kuwaas oo leh qaabab kiimiko oo kala duwan oo kor u qaadaya awoodda garashada iyo ka hortagga dhaawaca barashada iyo xusuusta iyada oo loo marayo saamaynta ay ku leeyihiin kiliyaha maskaxda.Ma laha sifooyinka muscarinic receptor agonists iyo antagonists, sidoo kale ma joojinayso dhaqdhaqaaqa Ach.Saamaynta ka-hortagga illowsiinta iyo xusuusta-kordhinta ee daawadan waxaa lagu gaaraa iyada oo la wanaajiyo sii-deynta Ach ee kiliyaha maskaxda.Kinases-ku-tiirsanaanta borotiinka waxay xoojisaa dhaqdhaqaaqa kanaalka Ca2+, kaas oo laga yaabo inay mas'uul ka yihiin sii dayntooda Ach.Nefiracetam (NEF) waa wakiilka nootropic ee nooca pyrrolidone oo leh dawooyin kala duwan iyo sidoo kale saamaynta kor u qaadista garashada.Qallalka amygdala-kindled, nefiracetam waxay joojisaa suuxdinta korantada iyo dabeecadda labadaba.NEF waxay leedahay spectrum anticonvulsant oo gooni ah.

Muuqaal

Nefiracetam waxaa loo isticmaalaa in lagu daaweeyo cudurrada maskaxda.Waxay kor u qaadi kartaa awoodda garashada waxayna ka hortagi kartaa dhaawaca barashada iyo xusuusta saamaynta ay ku leedahay kortex maskaxda.Ma laha sifooyinka muscarinic receptor agonist iyo wakiilka ka soo horjeeda, mana joojinayso dhaqdhaqaaqa acetyl cholinase.Sidaa darteed, saameynteeda ka-hortagga illowda iyo xusuusta-kor u qaadista waxay ku dhacdaa iyada oo hagaajinaysa sii-deynta acetylcholine ee kiliyaha maskaxda.

Codsiyada

Nefiracetam waa nooc ka mid ah hydrophobic of piracetam iyo synthesis synthetic ee dhammaan xeryahooda Racetam piracetam.Nefiracetam waxaa soo saaray ugu horrayn Daiichi Sankyo (shirkadda dawooyinka Japan) ee daaweynta AD.Marka lagu daro dhammaan hababka loo aaneeyo Nefiracetam, waxaa guud ahaan loo maleynayaa inay tahay walax ka masuul ah helitaanka kanaalada calcium ee jirka, iyo sidoo kale wareejinta aan tooska ahayn ee walaxda calaamadaynta kicinta, u dhaqma sida qayb ka mid ah agonist goobta glycine-ku-xidhida ee soo-dhoweeyaha NDMA.


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